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Search Results for " Gutathione S-transferase "

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4

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天然化合物

カタログ番号 製品名 別名 ターゲット
T11505 GSTO1-IN-1 Glutathione Peroxidase , GST
GSTO1-IN-1 is a potent glutathione S-transferase omega 1 inhibitor (GSTO1; IC50: 31 nM).
T5097 Ezatiostat TER199(free base),TLK199 Apoptosis , Glutathione Peroxidase , GST
Ezatiostat (TER199(free base)) is a tripeptide analog of glutathione that can selectively inhibit GSTP1-1 catalytic activity.
T4564 Ethacrynic acid Edecrin,Etacrynic Acid,Hydromedin Others , Calcium Channel , NF-κB , GST
Ethacrynic acid (Edecrin) is a nonsulfonamide loop diuretic that inhibits the activity of the Na+/K+/2Cl- cotransporter NKCC2 in the thick ascending limb of the loop of Henle. It also inhibits glutathione S-transferase a...
T22776 Ezatiostat hydrochloride TLK199 HCl,TER199 Glutathione Peroxidase
Ezatiostat hydrochloride (TLK199 HCl) is an effective inhibitor of glutathione S-transferase. Ezatiostat hydrochloride is a novel glutathione analog and the potential treatment of cytopenias. In addition, Ezatiostat hydr...
カタログ番号 製品名 別名 ターゲット
T3S0012 Coniferyl ferulate P-gp , GST
Coniferyl ferulate is a strong inhibitor of glutathione S-transferase (GST) isolated from Radix Angelicae sinensis. It shows strong inhibition of human placental GST (IC50: 0.3 μM). It also reverses multidrug resistance ...
TN1078 Seneciphylline P450 , GST
Seneciphylline, one of the hepatotoxic pyrolizidine alkaloids, has mutagenic activity in Drosophila and their transfer into rat milk.Seneciphylline can significantly increased the activities of epoxide hydrase and glutat...
T7995 α-Angelica lactone Alpha-Angelica Lactone Others , GST
α-Angelica lactone has cardiotonic activity, may exert their effects by providing an increased contraction-dependent calcium pool to be released upon systolic depolarization.
T3S0541 Curzerene Apoptosis , GST
Curzerene, a sesquiterpene compound derived from the rhizome of Curculigo orchioides Gaertn, possesses potent anti-cancer properties. It is known to induce apoptosis in cells[1] and also suppress the expression of glutat...